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Boc
Glaucarubin 1448
MCE
HA
MCE
FGL peptide 499993
trans Chlordane
YAP1 TFE3 mediates endothelial
SBI
JNJ
Functional Maturation of Cytochromes P4503A4 and 2D6 Relies on GAPDH
MCE
BMMSCs
164127
ZD0947 172649
Sema4d
AANAT
MCE
TLR7
DMTr
Basic yellow 28 54060
p
配对样同源域 2（PITX2）基因
Fenretinide glucuronide 79982
GS
TLR7 agonist 9
SK
Decyl decanoate 1654
hOR17
Design, Synthesis, and Antibacterial Activity of Novel Paeonol Derivatives Containing Piperazine Moiety PMID 41108272
含锚蛋白重复和 SOCS 框 9（ASB9）基因
chain
3,5
β
锌指蛋白 512B（ZNF512B）基因
SKP2 promotes the metastasis of pancreatic ductal adenocarcinoma by suppressing TRIM21
2
CTD 小磷酸酶 1（CTDSP1）基因
醋酸来法莫林
G 蛋白核仁 3 样（GNL3L）基因
BE2254 40077
MCE
GAP
YAP promotes multi
Cy3
含 Mab
Ligands for E3 Ligase
Amarogentin inhibits vascular smooth muscle cell proliferation and migration and attenuates neointimal hyperplasia via AMPK activation PMID 36906074
Vincristine Regulates C/EBP
The active GLP
lncRNA HOTAIR Promotes DNA Repair and Radioresistance of Breast Cancer via EZH2 PMID 33136445
Lupulone
Zopolrestat
Structure
transcription
Ozarelix
DMT
Epigenetic small molecule screening identifies a new HDACi compound for ameliorating Duchenne muscular dystrophy PMID 39974951
MCE
Antagonism of sigma
B16.F10
MCE
囊泡相关膜蛋白 2（VAMP2）基因
TC14012 368874
XST14
MCE
酪氨酰 DNA 磷酸二酯酶 1（TDP1）基因
Mixed Lineage Kinase
V116517 1073616
urinary tract infections
A
LEESGGGLVQPGGSMK 2096980
Genome
nude mouse
translocations
CP675206
富谷氨酰胺 1（QRICH1）基因
AC 7700
Decarbamoylmitomycin C
MCE
antiplasmin
Anti
Anti
126823
Anti
Staufen 抗体 (YA2077)（Staufen Antibody (YA2077)）
Rho GTP 酶激活蛋白 32（ARHGAP32）基因
高机动性组 20B（HMG20B）基因
Lipid Peroxide
线粒体核糖体蛋白 S18B（MRPS18B）基因
RSK1 is an exploitable dependency in myeloproliferative neoplasms and secondary acute myeloid leukemia PMID 39820365
FKBP52 抗体 (YA432)（FKBP52 Antibody (YA432)）
trachea
LRP2/Megalin 蛋白, Human (HEK293, His)
Novel adipokine asprosin modulates browning and adipogenesis in white adipose tissue PMID 33705351
Trienzymatic Complex System for Isomerization of Agar
Magnesium lithospermate B promotes proliferation and differentiation of neural stem cells in vitro and enhances neurogenesis in vivo PMID 30060831
P2Y12 antagonist 1
α
Fenhexamid
The metabolism of 3
Discovery of small molecule inhibitors of the PH domain leucine
THBS1
Etomoxir
MCE
FTY720 analogues as sphingosine kinase 1 inhibitors enzyme inhibition kinetics, allosterism, proteasomal degradation, and actin rearrangement in MCF
Trifloroside 53823
Asunercept 1450882
Cathepsin
Characterization of the metabolites of TUG
Ribosome
QL47B
(E/Z)
GA 结合蛋白转录因子亚基β2（GABPB2）基因
2
阿比多尔盐酸盐
influx,nitrobenzylthioinosine
Degradation products of cyanidin glycosides from tart cherries and their bioactivities PMID 11600045
Anti
Ribosomal S6 Kinase (RSK)
translocation
Olaparib Enhances the Efficacy of Third
MCE
Characterization of a HIR
Matrix metalloproteinases
HMGB1
ADAM12
RCN2 facilitates esophageal squamous cellular carcinoma metastasis and cisplatin resistance through UBR5
Inhibition of kynurenine aminotransferase II reduces activity of midbrain dopamine neurons PMID 26514401
DUBs
urinary tract infections
The ribosomal S6 kinase inhibitor BI
Oncolytic adenovirus delivery of neoantigens sensitizes low
Sirtuin
Oligonuclear polypyridylruthenium(II) complexes incorporating flexible polar and non
cell cycle
Anti
艾尔骨化醇
Anti
MB
芹菜素
Propargyl
Polyphenol and glucosinolate
fucose oligosaccharide
Zinc chloride, meets analytical specification of Ph. Eur. BP USP
Anti
NOC 18
suppressor
睾丸表达 11（TEX11）基因
FGFR
Ca channels
Candidone
S
SIRT7 抗体 (YA6765)（SIRT7 Antibody (YA6765)）
SID
I
马来酸氨氯地平
1,2,3,4,6
Exosomal lipid PI4P regulates small extracellular vesicle secretion by modulating intraluminal vesicle formation PMID 37021404
Atractylodin Induces Apoptosis and Inhibits the Migration of A549 Lung Cancer Cells by Regulating ROS
Effect of ranirestat, a new aldose reductase inhibitor, on diabetic retinopathy in SDT rats PMID 25215304
Blood glucose regulation
Securinine, a myeloid differentiation agent with therapeutic potential for AML PMID 21731671
Berberine chloride 633
Classical swine fever virus infection suppresses claudin
Methyl diethyldithiocarbamate
Discovery of New Monocarbonyl Ligustrazine
Phytosterol
Pentamidine is an antiparasitic and apoptotic drug that selectively modifies ubiquitin PMID 17191940
Activation of TGR5 protects blood brain barrier via the BRCA1/Sirt1 pathway after middle cerebral artery occlusion in rats PMID 32381096
GSH exhaustion via inhibition of xCT
Valnoctamide, valpromide and valnoctic acid are much less teratogenic in mice than valproic acid PMID 9551843
Sirtuin
SIRP alpha/CD172a 蛋白, Human (119a.a, HEK293, Llama Fc)
Fate of primary cells at the G₁/S boundary after polo
5
HGF/c
SOS1
Synthesis of novel hybrid quinolino[4,3
modulator
Identification of galectin
Hyperactivity of Hypothalamic
Tioxaprofen 40198
Anti
Aspartoacylase suppresses prostate cancer progression by blocking LYN activation PMID 37271807
PAX6 抗体(YA6612)（PAX6 Antibody(YA6612)）
Anti
Aspergillumarin B
IQTub4P
Calcium Channel antagonist 5
A 1335
Glucametacine
[Ala92]
沉默信息调节因子 2 相关酶类 7（SIRT7）基因
Anti
CYP1B1
Chloroquine
Anti
bladder
3'
Ru(bpy)2(mcbpy
CD94 蛋白, Human (HEK293, His)
Aberrant MCM10 SUMOylation induces genomic instability mediated by a genetic variant associated with survival of esophageal squamous cell carcinoma PMID 34185429
Bardoxolone
epigenetic
A549 cells
Carbasalate calcium (卡巴匹林钙)
Anti
brain
AG 3340
Resmethrin (Benzofuroline)
Anti
ULK
Anti
K201 (JTV519) is a Ca2+
Picrotoxinin 17617
MCE
Liothyronine
FGL2 蛋白, Human (HEK293, His
DYRK1A
The ARID1A
The antipsychotic drug thiothixene stimulates macrophages to clear pathogenic cells by inducing arginase 1 and continual efferocytosis PMID 40198748
YS
N,N'
4
Biotin
1C 型激活素 A 受体（ACVR1C）基因
Effects of BAMBI on luteinized follicular granulosa cell proliferation and steroid hormone production in sheep PMID 36775976
Discovery of a novel quinoxaline derivative modulator via a dual P53/TLR2 targeting strategy for the alleviation of radiation damage PMID 40112665
Antibacterial effect of caprylic acid and monocaprylin on major bacterial mastitis pathogens PMID 16162522
Multicomponent Synthesis of 2,4,5
DNA glycosylases provide antiviral defence in prokaryotes PMID 38632404
(
TYMS 反链 RNA（TYMSOS）基因
Synthesis, activity, and pharmacophore development for isatin
Radiation induces ESCRT pathway dependent CD44v3+ extracellular vesicle production stimulating pro
An exploration of the protective effects of Ginsenoside Rb1 against acute lung injury using network pharmacology, molecular docking, molecular dynamics simulations, and in vivo experiments PMID 40347881
The antihypertensive drug hydralazine activates the intrinsic pathway of apoptosis and causes DNA damage in leukemic T cells PMID 26942461
Chemistry of clothianidin and related compounds PMID 20873771
Triapine hydrochloride 216240
毛叶长春花提取物 (Catharanthus trichophyllus (Baker) Pichon)
Identifying the mechanisms underlying the protective effect of tetramethylpyrazine against cisplatin‑induced in vitro ototoxicity in HEI‑OC1 auditory cells using gene expression profiling PMID 33174043
SMIP004 143360
LRRK2 抗体 (YA2821)（LRRK2 Antibody (YA2821)）
[A clinical study on lamivudine treatment for advanced schistosomisis with chronic B hepatits] PMID 24490380
LncRNA SNHG14 promotes hepatocellular carcinoma progression via H3K27 acetylation activated PABPC1 by PTEN signaling PMID 32811821
Dapagliflozin attenuates diabetes
Lixisenatide, a drug developed to treat type 2 diabetes, shows neuroprotective effects in a mouse model of Alzheimer's disease PMID 25107586
HSP105 suppresses the progression of cutaneous squamous cell carcinoma by activating the P53 signaling pathway PMID 37559974
The serotonin(5
1,2,3
Ro 67
Rhamnetin and cirsiliol induce radiosensitization and inhibition of epithelial
Quantification of the irreversible fibroblast growth factor receptor inhibitor futibatinib by UPLC
JT001 sodium 2238820
Structure
GZD856 (formic) 2804039
Lynamicin B is a Potential Pesticide by Acting as a Lepidoptera
Membrane RRM2
(S)
Tectorigenin alleviates intrahepatic cholestasis by inhibiting hepatic inflammation and bile accumulation via activation of PPARγ PMID 33661551
Conformational flexibility and inhibitor binding to unphosphorylated interleukin
Hydroxy
Electrophysiological evidence showing muscarinic agonist
Characterization of raloxifene glucuronidation in vitro contribution of intestinal metabolism to presystemic clearance PMID 12019197
m
Emodin facilitates the transformation of A1/A2 reactive astrocytes through the 11β
Antibacterial agent 219
Physalis Calyx seu Fructus inhibited pulmonary fibrosis through regulating Wnt/β
Human T Helper 9 Cells Rely on Peroxisome Proliferator
The Effect of Piperine Pro
NH
Ligustroflavone reduces necroptosis in rat brain after ischemic stroke through targeting RIPK1/RIPK3/MLKL pathway PMID 31055628
A New Spin on Antibody
MMA
(S)
5
Exposure to polystyrene microplastics causes reproductive toxicity through oxidative stress and activation of the p38 MAPK signaling pathway PMID 31896473
Involvement of glutamate NMDA and AMPA receptors, glial cells and IL
A phase 1 study of LY3076226, a fibroblast growth factor receptor 3 (FGFR3) antibody
L
Inhibitory effects of schisandrin A and schisandrin B on CYP3A activity PMID 20448858
1
Application of newly developed and validated UPLC
Telocinobufagin, a Novel Cardiotonic Steroid, Promotes Renal Fibrosis via Na⁺/K⁺
7
1
辅酶 Q9（COQ9）基因
Siweixizangmaoru Decoction Ameliorated Type II Collagen
Two new 14, 15
Chemotherapeutic agent CPT
Atractylenolide I restores HO
Caspase
LncRNA HOXB
Pilocarpine
Bacteria escape macrophage
DDX24 promotes tumor progression by mediating hexokinase
Species
Safimaltib 2230273
5
Implementation of toxicokinetics in toxicity studies
N
IL
Valdecoxib
Indobufen 63610
2
D
MDL 29913 135721
Amino
4,6
The nasal decongestant effect of xylometazoline in the common cold PMID 18655753
Cantharidic acid 28874
L
Sporminarin B 915403
Anti
ML329 19992
溶质载体家族 39 成员 1（SLC39A1）基因
Hippocampal CaMKII inhibition induces reactivation
Futoamide 23477
GW 766994 408303
D
Ms
EGFR/Cytokine
TAMRA
CD276
A novel mGluR5 antagonist, MFZ 10
TCS 183
Rho 鸟嘌呤核苷酸交换因子 1（ARHGEF1）基因
(2
Technical Support
(2S,3AS,7aS)
Nodosin 10391
Characterization of a dual degrader of MDM2 and GSPT1 PMID 40440791
Rescuing SERCA2 pump deficiency improves bone mechano
Alpha2A
1
Kaempferol attenuates wear particle
CTCE
In Vivo Antistress Effects of Synthetic Flavonoids in Mice Behavioral and Biochemical Approach PMID 35209189
Tenovin
Suramin ameliorates osteoarthritis by acting on the Nrf2/HO
C
Natural Oncolysis of Enterovirus 71 in Antitumor Therapy of Colorectal Cancer PMID 37132155
L1CAM 蛋白, Human (HEK293, His, solution)
DHRS13 suppresses differentiation and mitophagy in glioma via retinoic acid and mitochondrial reactive oxygen species PMID 40739132
Ibuprofen sodium 31121
Elucidating the molecular pharmacology of trace amine
m
Lucanthone and its derivative hycanthone inhibit apurinic endonuclease
Arachidonic acid 506
Discovery of novel allosteric modulators of metabotropic glutamate receptor subtype 5 reveals chemical and functional diversity and in vivo activity in rat behavioral models of anxiolytic and antipsychotic activity PMID 20923853
HGF
Low
SIRP alpha V6/CD172a 蛋白, Human (Biotinylated, HEK293, His
1
Daily voluntary exercise enhances pilocarpine
Intraplantar β
4
1
Regulation of kainate receptors by cAMP
4
Novel merosesquiterpene exerts a potent antitumor activity against breast cancer cells in vitro and in vivo PMID 24704691
Amphotericin B encapsulated in micelles based on poly(ethylene oxide)
Design and synthesis of novel 1,2,3
Keratin sulfate 169799
On the mode of action of 7
ExoSTING, an extracellular vesicle loaded with STING agonists, promotes tumor immune surveillance PMID 33888863
Intracellular AIBP (Apolipoprotein A
Octylbenzene
First comprehensive structural and biophysical analysis of MAPK13 inhibitors targeting DFG
Antioxidant and anti
Receptor affinities of dopamine D1 receptor
Inhibition of TRPP3 channel by amiloride and analogs PMID 17804601
干扰素λ受体 1（IFNLR1）基因
S
E3 ubiquitin ligase CHIP facilitates cAMP and cGMP signalling cross
2,4
The integrin repertoire drives YAP
Targeting OXPHOS de novo purine synthesis as the nexus of FLT3 inhibitor
t
Antibacterial mechanism of allyl isothiocyanate PMID 10852565
RAP
Tislelizumab 1858168
Verbascoside Alleviates Atopic Dermatitis
Initial testing (stage 1) of the BH3 mimetic ABT
TDPAM01
Corosolic acid sensitizes ferroptosis by upregulating HERPUD1 in liver cancer cells PMID 36038536
MEY
Walnut oil alleviates LPS
ENPP
Substrate
Functional Characterization of an Arylsulfonamide
pH
Large
PFKP facilitates ATG4B phosphorylation during amino acid deprivation
N
Synthesis and antiviral evaluation of acyclic azanucleosides developed from sulfanilamide as a lead structure PMID 18778942
BCL2 相关的细胞死亡激动因子（BAD）基因
Sarcosine
p38 kinase inhibitors for the treatment of arthritis and osteoporosis thienyl, furyl, and pyrrolyl ureas PMID 11140741
Metabolic effects of insulin blockade by D
C1q
VU590
PLK1/BRD4
Sch 40853
Ethyl 2
Development of a High
Transcriptomics and metabolomics reveal changes in the regulatory mechanisms of osteosarcoma under different culture methods in vitro PMID 36536381
Long non
Propargyl
蛋白酶体 26S 亚基，ATPase 1（PSMC1）基因
Novel inhibition of PIM2 kinase has significant anti
Medical therapy to attenuate fetal anaemia in severe maternal red cell alloimmunisation PMID 32794242
Cletoquine
Pizotifen (Pizotyline，苯噻啶)
Effects of ketoprofen, morphine, and kappa opioids on pain
磷酸二酯酶 6G（PDE6G）基因
Acid
Lienal Polypeptide Decreases Immune Thrombocytopenia in a Mouse Model by Upregulating Cytokine Production and Increasing the Levels of CD4+, CD8+, and T Regulatory Cells PMID 40113259
Ag2S
The structural basis for the phospholipid remodeling by lysophosphatidylcholine acyltransferase 3 PMID 34824256
2,4,6
含 pleckstrin 同源结构域 N1（PLEKHN1）基因
RAR/RXR
Protective Actions of Epithelial 5
20
IL
Enhanced Myogenesis by Silencing Myostatin with Nonviral Delivery of a dCas9 Ribonucleoprotein Complex PMID 35758824
Peptidyl anthraquinones as potential antineoplastic drugs synthesis, DNA binding, redox cycling, and biological activity PMID 8759632
Felodipine induces autophagy in mouse brains with pharmacokinetics amenable to repurposing PMID 31000720
Mesenchymal Stem Cell
卡林 3（CUL3）基因
Styrene
5
Near
Ethacrynic acid a novel radiation enhancer in human carcinoma cells PMID 8567338
CD38 inhibitor 2 2597933
HY
D
Loss of DNA Polymerase β Delays Atherosclerosis in ApoE
LPS enhances platelets aggregation via TLR4, which is related to mitochondria damage caused by intracellular ROS, but not extracellular ROS PMID 29653689
Nomegestrol acetate 58652
SVM model for virtual screening of Lck inhibitors PMID 19267483
Equilin in conjugated equine estrogen increases monocyte
Tetraethylene glycol monohexadecyl ether 5274
3
Alvespimycin hydrochloride 467214
The effect of celecoxib on tumor growth in ovarian cancer cells and a genetically engineered mouse model of serous ovarian cancer PMID 27074576
华中五味子提取物 (Schisandra sphenanthera Rehd. et Wils)
Structural and functional characterization of HQL
8
inhibitor
MEK
Co
CD20
AZ1495 2196204
Dacarbazine
Synthesis, biological evaluation and molecular modeling of novel azaspiro dihydrotriazines as influenza virus inhibitors targeting the host factor dihydrofolate reductase (DHFR) PMID 29886325
PNT6555
[Detection and identification of new pungent compounds in fruits of Capsicum (author's transl)] PMID 461555
Selective inhibition of cocaine
Rational Design of Highly Potent SARS
Structure
Differential effects of etifoxine on anxiety
The loss of B7
DAPK enhances DDX20 protein stability via suppression of TRIM25
Methyl 10(S),11(S)
Carbohydrate Sulfotransferase 1 (EC 2.8.2.21)
17
Arformoterol 67346
5’
Benzyl
Liraglutide 204656
Differential enzymatic characteristics and tissue
A hippocampus dependent neural circuit loop underlying the generation of auditory mismatch negativity PMID 35026286
Cancer associated fibroblast
SAMHD1 Limits the Efficacy of Forodesine in Leukemia by Protecting Cells against the Cytotoxicity of dGTP PMID 32402273
Effects of local administration of tiludronic acid on experimental periodontitis in diabetic rats PMID 28914593
ANGPTL3/Angiopoietin
High Affinity Binding of N2
Methylthiomcresol
Silencing of activin receptor
Peptide Hydrogels as Immunomaterials and Their Use in Cancer Immunotherapy Delivery PMID 37256647
3’
Ethyl pyruvate administration inhibits hepatic tumor growth PMID 19584311
Simultaneous Semimechanistic Population Analyses of Levofloxacin in Plasma, Lung, and Prostate To Describe the Influence of Efflux Transporters on Drug Distribution following Intravenous and Intratracheal Administration PMID 26621623
IL
Nivalenol 23282
TRIM21 Promotes Oxidative Stress and Ferroptosis through the SQSTM1
Disulfiram
Haloperidol
AG2034 177575
Inhibition of glycogen synthase kinase
Anti
Peptide
Antioxidant, antiradical, and anticholinergic properties of cynarin purified from the Illyrian thistle (Onopordum illyricum L.) PMID 25792498
Butyrylcarnitine
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